GPCR Target Tracking & Status
Success
In Progress Collaborator Progress Failed Work Stopped
|
GPCR Net ID |
Protein Name |
Uniprot |
Ligand/Lattice |
Cloning |
Expression |
Purification |
Crystallization |
Diffraction |
Structure |
Refinement |
PDB |
|
1* |
5-hydroxytryptamin
(serotonin) receptor 1A |
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2 |
5-hydroxytryptamin
(serotonin) receptor 2C |
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4 |
5-hydroxytryptamine
receptor 2B |
Ergotamine |
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6 |
adenosine A2a
receptor |
ZM241385 |
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UK-432097 |
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ZM241385 (1.8 Ang) |
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11* |
Angiotensin II
receptor 1 |
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15 |
beta-2-adrenergic
receptor |
Carazolol |
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Timolol |
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Alprenolol |
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ICI 118,551 |
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Compound1 |
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16 |
beta-3-adrenergic
receptor |
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17* |
Blue sensitive opsin |
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25 |
cannabinoid
receptor 1 (CB1) |
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27U |
CCR1 |
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28*U |
CCR5 |
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31U |
CXCR1 |
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32U |
CXCR2 |
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33*U |
CXCR3 |
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34*U |
CXCR4 |
|
CVX15 |
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IT1t |
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IT1t (I222) |
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IT1t (P1) |
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IT1t (P1) |
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36 |
D1 dopamine
receptor |
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38 |
D3 dopamine
receptor |
Eticlopride |
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39* |
delta opioid
receptor |
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48 |
Ghrelin receptor |
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49 |
Glucagon receptor
(GLR) |
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50 |
Glucose-dependent insulinotropic receptor |
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51* |
Gonadotropin-releasing
hormone receptor |
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53 |
Histamine receptor
H1 |
Doxepin |
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56* |
kappa opioid
receptor |
JDTic |
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65 |
Melanocortin 4 receptor |
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68 |
Metabotropic
glutamate receptor 1 |
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71* |
mu opioid receptor |
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74 |
Neurokinin 1 receptor
(Substance P receptor) |
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79* |
nociceptin opioid
receptor (ORL-1) |
Compound-24 |
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|
80 |
Olfactory receptor
1A1 |
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87 |
P2Y purinoceptor 12 |
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90 |
Prostaglandin E2
receptor EP2 subtype |
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93* |
Proteinase-activated receptor 1 |
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110 |
Sphingosine 1-phosphate receptor 1 |
ML056 |
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118* |
5-hydroxytryptamine
receptor 1B |
dihydroergotamine |
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ergotamine |
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119 |
Olfactory receptor
51L1 |
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120 |
Olfactory receptor
10A6 |
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121 |
Olfactory receptor
2A25 |
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122 |
Olfactory receptor
5K1 |
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123* |
Red-sensitive opsin |
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124* |
Green-sensitive opsin |
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125* |
Parathyroid hormone
1 receptor |
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126* |
Corticotropin-releasing factor
receptor 1 |
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127* |
PACAP-R1 |
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128 |
Metabotropic
glutamate receptor 4 |
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129 |
Metabotropic
glutamate receptor 5 |
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130 |
Metabotropic glutamate
receptor 7 |
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131 |
Smoothened Receptor |
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*Entries are Community Nominated
Targets, UEntries are U01 Targets, Targets are being
pursued with collaborators